Inhibition of the lipolytic action of beta-adrenergic agonists in human adipocytes by alpha-adrenergic agonists.
نویسندگان
چکیده
منابع مشابه
Beta-Adrenergic Agonists
Inhaled β₂-adrenoceptor (β₂-AR) agonists are considered essential bronchodilator drugs in the treatment of bronchial asthma, both as symptoms-relievers and, in combination with inhaled corticosteroids, as disease-controllers. In this article, we first review the basic mechanisms by which the β₂-adrenergic system contributes to the control of airway smooth muscle tone. Then, we go on describing ...
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Incubation of human distal bronchi from 48 patients for 15 h with 10(-7) M fenoterol induced sensitization characterized by an increase in maximal contraction to endothelin-1 (ET-1) and acetylcholine (ACh). Incubation of human bronchi with 10(-6), 3 x 10(-6), and 10(-5) M forskolin (an adenyl cyclase activator) reproduced sensitization to ET-1 and ACh. The sensitizing effect of fenoterol was in...
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CHRISTOPHE FAISY,1,2 EMMANUEL NALINE,1 JEAN-LUC DIEHL,2 XAVIER EMONDS-ALT,3 THIERRY CHINET,1 AND CHARLES ADVENIER1 1Unité Propre de Recherche de l’Enseignement Supérior Equipe d’Accueil 220, Faculté de Médecine Paris-Ouest, Unité de Formation et de Recherche Biomédicale des Saint-Pères, 75006 Paris; 2Service de Réanimation Médicale, Hôpital Européen Georges Pompidou, 75908 Paris Cedex 15; and 3...
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ژورنال
عنوان ژورنال: Journal of Lipid Research
سال: 1981
ISSN: 0022-2275
DOI: 10.1016/s0022-2275(20)37319-3